Vitamin D receptor (VDR) agonist
Prodrug of vitamin D3.
Vitamin D2 analog, VDR agonist.
Vitamin D3 analog.
Potent inhibitor of aurora kinases with Ki values to be 0.6, 18 and 4.6 nM for auraro A, B and C isotypes respectively.
Prohormone of calcitriol. Major circulating form of vitamin D.
Potent, reversible AMP-activated protein kinase (AMPK) activator.
(+)-Bicuculline is an antagonist of the GABAA receptor.
CYC116 (CYC-116)is an oral small molecule Aurora kinase/VEGFR2 inhibitor with antineoplastic activity.
Potent D3 dopamine receptor agonist (Ki = 2.3 nM).
A potent and specific Aurora kinase B inhibitor
P-glycoprotein (P-gp) modulator; inhibits P-gp-mediated multidrug-resistance (MDR).
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