Products List
More detailed classification
mTOR     PI3K   

Dual kinase inhibitor; inhibits PI 3K family kinases.
GDC-0941 is an orally bioavailable bismesylate salt of a potent small-molecule thieno[3,2-d]pyrimidine inhibitor.
BEZ235 (NVP-BEZ235) is an inhibitor of PI3K and mTOR.p110, IC50<6nM.
A66 is a highly specific and selective p110α inhibitor with IC50 of 32,30 and 43 nM for p110α, p110α/E545K, p110α/E545K, p110α/H1047R, respectively.
A potent inhibitor of PI 3-kinase activity, acting as a competitive inhibitor for ATP binding site of the enzyme.
Potent and selective mTOR inhibitor (IC50 = 2.1 nM).
Potent and selective mTOR inhibitor (IC50 = 2 - 10 nM for mTORC1 and mTORC2).
PP242 has been shown to be a potent and selective mTOR inhibitor.
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